GENERAL ORGANIC CHEMISTRY
Lin L, Patel EN, Nielsen AL, Turner LD, Tepp WH, Nguyen K, Pellett S, Janda K. Transformation of a metal chelate into a “catch and anchor” inhibitor of Botulinum A protease. Int J Mol Sci. 2023;24(5). PMID: 36901734.
Patel EN, Lin L, Sneller MM, Eubanks LM, Tepp WH, Pellett S, Janda KD. Investigation of salicylanilides as botulinum toxin antagonists. ACS Infect Dis. 2022;8(8):1637-45. PMID: 35877209.
Blake S, Shaabani N, Eubanks LM, Maruyama J, Manning JT, Beutler N, Paessler S, Ji H, Teijaro JR, Janda KD. Salicylanilides reduce SARS-CoV-2 replication and suppress induction of inflammatory cytokines in a rodent model. ACS Infect Dis. 2021;7(8):2229-37. PMID: 34339171.
Natori Y, Kim D J. Synthesis of drug vaccine against heroin contaminated with fentanyl and their biological evaluation. J Synth Org Chem Jpn. 2020;78(9):875-85.
Kimishima A, Olson ME, Natori Y, Janda KD. Efficient syntheses of cocaine vaccines and their in vivo evaluation. ACS Med Chem Lett. 2018;9(5):411-6. PMID: 29795751.
Miranda PO, Cubitt B, Jacob NT, Janda KD, de la Torre JC. Mining a Kröhnke pyridine library for anti-arenavirus activity. ACS Infect Dis. 2018;4(5):815-24. PMID: 29405696.
Anraku K, Sato S, Jacob NT, Eubanks LM, Ellis BA, Janda KD. The design and synthesis of an alpha-Gal trisaccharide epitope that provides a highly specific anti-Gal immune response. Org Biomol Chem. 2017;15(14):2979-92. PMID: 28294277.
Srinivasulu V, Janda KD, Abu-Yousef IA, O'Connor MJ, Al-Tel TH. A modular CuI-L-proline catalyzed one-pot route for the rapid access of constrained and privileged hetero-atom-linked medium-sized ring systems. Tetrahedron. 2017;73(15):2139-50.
Cai X, Janda KD. A chemoenzymatic approach toward the preparation of site-specific antibody–drug conjugates. Tetrahedron Lett. 2015;56(23):3172-5.
Seki H, Pellett S, Silhar P, Stowe GN, Blanco B, Lardy MA, Johnson EA, Janda KD. Synthesis/biological evaluation of hydroxamic acids and their prodrugs as inhibitors for Botulinum neurotoxin A light chain. Bioorg Med Chem. 2014;22(3):1208-17. PMID: 24360826.
Fullagar JL, Garner AL, Struss AK, Day JA, Martin DP, Yu J, Cai X, Janda KD, Cohen SM. Antagonism of a zinc metalloprotease using a unique metal-chelating scaffold: Tropolones as inhibitors of P. aeruginosa elastase. Chem Commun (Camb). 2013;49(31):3197-9. PMID: 23482955.
Silhar P, Eubanks LM, Seki H, Pellett S, Javor S, Tepp WH, Johnson EA, Janda KD. Targeting botulinum A cellular toxicity: A prodrug approach. J Med Chem. 2013;56(20):7870-9. PMID: 24127873.
Garner AL, Gloeckner C, Tricoche N, Zakhari JS, Samje M, Cho-Ngwa F, Lustigman S, Janda KD. Design, synthesis, and biological activities of closantel analogues: Structural promiscuity and its impact on Onchocerca volvulus. J Med Chem. 2011;54(11):3963-72. PMID: 21534605.
Garner AL, Yu J, Struss AK, Lowery CA, Zhu J, Kim SK, Park J, Mayorov AV, Kaufmann GF, Kravchenko VV, Janda KD. Synthesis of 'clickable' acylhomoserine lactone quorum sensing probes: Unanticipated effects on mammalian cell activation. Bioorg Med Chem Lett. 2011;21(9):2702-5. PMID: 21190852.
Moreno AY, Mayorov AV, Janda KD. Impact of distinct chemical structures for the development of a methamphetamine vaccine. J Am Chem Soc. 2011;133(17):6587-95. PMID: 21473576.
Silhar P, Alakurtti S, Capkova K, Xiaochuan F, Shoemaker CB, Yli-Kauhaluoma J, Janda KD. Synthesis and evaluation of library of betulin derivatives against the botulinum neurotoxin A protease. Bioorg Med Chem Lett. 2011;21(8):2229-31. PMID: 21421315.
Stowe GN, Janda KD. A Diels-Alder reaction conducted within the parameters of aqueous organocatalysis: Still just smoke and mirrors. Tetrahedron Lett. 2011;52(17):2085-7. PMID: 21516231.
Zakhari JS, Kinoyama I, Hixon MS, Di Mola A, Globisch D, Janda KD. Formulating a new basis for the treatment against botulinum neurotoxin intoxication: 3,4-diaminopyridine prodrug design and characterization. Bioorg Med Chem. 2011;19(21):6203-9. PMID: 21975066.
Capkova K, Hixon MS, Pellett S, Barbieri JT, Johnson EA, Janda KD. Benzylidene cyclopentenediones: First irreversible inhibitors against botulinum neurotoxin A's zinc endopeptidase. Bioorg Med Chem Lett. 2010;20(1):206-8. PMID: 19914829.
Silhar P, Capkova K, Salzameda NT, Barbieri JT, Hixon MS, Janda KD. Botulinum neurotoxin A protease: Discovery of natural product exosite inhibitors. J Am Chem Soc. 2010;132(9):2868-9. PMID: 20158239.
Frederick MO, De Lamo Marin S, Janda KD, Nicolaou KC, Dickerson TJ. Monoclonal antibodies with orthogonal azaspiracid epitopes. ChemBioChem. 2009;10(10):1625-9. PMID: 19492388.
Sheng J, Oyler G, Zhou B, Janda K, Shoemaker CB. Identification and characterization of a novel cell-penetrating peptide. Biochem Biophys Res Commun. 2009;382(2):236-40. PMID: 19084505.
Debler EW, Kaufmann GF, Meijler MM, Heine A, Mee JM, Pljevaljcic G, Di Bilio AJ, Schultz PG, Millar DP, Janda KD, Wilson IA, Gray HB, Lerner RA. Deeply inverted electron-hole recombination in a luminescent antibody-stilbene complex. Science. 2008;319(5867):1232-5. PMID: 18309081.
Richardson HN, Zhao Y, Fekete EM, Funk CK, Wirsching P, Janda KD, Zorrilla EP, Koob GF. MPZP: A novel small molecule corticotropin-releasing factor type 1 receptor (CRF1) antagonist. Pharmacol Biochem Behav. 2008;88(4):497-510. PMID: 18031798.
Willis B, Eubanks LM, Wood MR, Janda KD, Dickerson TJ, Lerner RA. Biologically templated organic polymers with nanoscale order. Proc Natl Acad Sci U S A. 2008;105(5):1416-9. PMID: 18216240.
Debler EW, Kaufmann GF, Kirchdoerfer RN, Mee JM, Janda KD, Wilson IA. Crystal structures of a quorum-quenching antibody. J Mol Biol. 2007;368(5):1392-402. PMID: 17400249.
Ino A, Dickerson TJ, Janda KD. Positional linker effects in haptens for cocaine immunopharmacotherapy. Bioorg Med Chem Lett. 2007;17(15):4280-3. PMID: 17531484.
McAllister LA, Hixon MS, Schwartz R, Kubitz DS, Janda KD. Synthesis and application of a novel ligand for affinity chromatography based removal of endotoxin from antibodies. Bioconjug Chem. 2007;18(2):559-66. PMID: 17315943.
Xu Y, Hixon MS, Dawson PE, Janda KD. Development of a FRET assay for monitoring of HIV gp41 core disruption. J Org Chem. 2007;72(18):6700-7. PMID: 17685571.
Boldt GE, Dickerson TJ, Janda KD. Emerging chemical and biological approaches for the preparation of discovery libraries. Drug Discov Today. 2006;11(3-4):143-8. PMID: 16533712.
Brogan AP, Dickerson TJ, Janda KD. Enamine-based aldol organocatalysis in water: Are they really "all wet"? Angew Chem Int Ed Engl. 2006;45(48):8100-2. PMID: 17001595.
Kim Y, Lillo AM, Steiniger SC, Liu Y, Ballatore C, Anichini A, Mortarini R, Kaufmann GF, Zhou B, Felding-Habermann B, Janda KD. Targeting heat shock proteins on cancer cells: Selection, characterization, and cell-penetrating properties of a peptidic GRP78 ligand. Biochemistry. 2006;45(31):9434-44. PMID: 16878978.
Moss JA, Stokols S, Hixon MS, Ashley FT, Chang JY, Janda KD. Solid-phase synthesis and kinetic characterization of fluorogenic enzyme-degradable hydrogel cross-linkers. Biomacromolecules. 2006;7(4):1011-6. PMID: 16602715.
Rogers CJ, Dickerson TJ, Janda KD. Kinetic isotope and thermodynamic analysis of the nornicotine-catalyzed aqueous aldol reaction. Tetrahedron. 2006;62(2):352-6.
Shigenaga A, Moss JA, Ashley FT, Kaufmann GF, Janda KD. Solid-phase synthesis and cyclative cleavage of quorum sensing depsipeptide analogues by acylphenyldiazene activation. Synlett. 2006;2006(4):0551-4.
Xu Y, Lu H, Kennedy JP, Yan X, McAllister LA, Yamamoto N, Moss JA, Boldt GE, Jiang S, Janda KD. Evaluation of "credit card" libraries for inhibition of HIV-1 gp41 fusogenic core formation. J Comb Chem. 2006;8(4):531-9. PMID: 16827565.
Xu Y, Shi J, Yamamoto N, Moss JA, Vogt PK, Janda KD. A credit-card library approach for disrupting protein-protein interactions. Bioorg Med Chem. 2006;14(8):2660-73. PMID: 16384710.
Zhang L, Long H, Boldt GE, Janda KD, Schatz GC, Lewis FD. α- and β-stilbenosides as base-pair surrogates in DNA hairpins. Org Biomol Chem. 2006;4(2):314-22. PMID: 16391774.
Dickerson TJ, Janda KD. Recent advances for the treatment of cocaine abuse: Central nervous system immunopharmacotherapy. AAPS J. 2005;7(3):E579-86. PMID: 16353936.
Kaufmann GF, Meijler MM, Sun C, Chen DW, Kujawa DP, Mee JM, Hoffman TZ, Wirsching P, Lerner RA, Janda KD. Enzymatic incorporation of an antibody-activated blue fluorophore into DNA. Angew Chem Int Ed Engl. 2005;44(14):2144-8. PMID: 15742317.
Lee BS, Mahajan S, Janda KD. Molecular iodine-catalyzed imine activation for three-component nucleophilic addition reactions. Synlett. 2005;2005(08):1325-7.
Lee BS, Mahajan S, Janda KD. Asymmetric dihydroxylation catalyzed by ionic polymer-supported osmium tetroxide. Tetrahedron Lett. 2005;46(26):4491-3.
Lee BS, Mahajan S, Janda KD. Cross-linked poly(4-vinylpyridine/styrene) copolymers as a support for immobilization of ytterbium triflate. Tetrahedron. 2005;61(12):3081-6.
Lee BS, Mahajan S, Janda KD. Novel method for catalyst immobilization using an ionic polymer: A case study using recyclable ytterbium triflate. Tetrahedron Lett. 2005;46(5):807-10.
Qi L, Yamamoto N, Meijler MM, Altobell LJ, 3rd, Koob GF, Wirsching P, Janda KD. △9-tetrahydrocannabinol immunochemical studies: Haptens, monoclonal antibodies, and a convenient synthesis of radiolabeled delta9-tetrahydrocannabinol. J Med Chem. 2005;48(23):7389-99. PMID: 16279798.
Reed NN, Dickerson TJ, Boldt GE, Janda KD. Enantioreversal in the Sharpless asymmetric epoxidation reaction controlled by the molecular weight of a covalently appended achiral polymer. J Org Chem. 2005;70(5):1728-31. PMID: 15730294.
Rogers CJ, Mee JM, Kaufmann GF, Dickerson TJ, Janda KD. Toward cocaine esterase therapeutics. J Am Chem Soc. 2005;127(28):10016-7. PMID: 16011362.
Rogers CJ, Dickerson TJ, Brogan AP, Janda KD. Hammett correlation of nornicotine analogues in the aqueous aldol reaction: Implications for green organocatalysis. J Org Chem. 2005;70(9):3705-8. PMID: 15845010.
Shimomura O, Se Lee B, Meth S, Suzuki H, Mahajan S, Nomura R, Janda KD. Synthesis and application of polytetrahydrofuran-grafted polystyrene (PS–PTHF) resin supports for organic synthesis. Tetrahedron. 2005;61(51):12160-7.
Shute TS, Matsushita M, Dickerson TJ, La Clair JJ, Janda KD, Burkart MD. A site-specific bifunctional protein labeling system for affinity and fluorescent analysis. Bioconjug Chem. 2005;16(6):1352-5. PMID: 16287229.
Yamashita M, Lee S-H, Koch G, Zimmermann J, Clapham B, Janda KD. Solid-phase synthesis of oxazolones and other heterocycles via Wang resin-bound diazocarbonyls. Tetrahedron Lett. 2005;46(33):5495-8.
Dickerson TJ, Lovell T, Meijler MM, Noodleman L, Janda KD. Nornicotine aqueous aldol reactions: Synthetic and theoretical investigations into the origins of catalysis. J Org Chem. 2004;69(20):6603-9. PMID: 15387581.
Kim YS, Moss JA, Janda KD. Biological tuning of synthetic tactics in solid-phase synthesis: Application to Aβ(1-42). J Org Chem. 2004;69(22):7776-8. PMID: 15498016.
Lee BS, Mahajan S, Clapham B, Janda KD. Suspension ring-opening metathesis polymerization: The preparation of norbornene-based resins for application in organic synthesis. J Org Chem. 2004;69(10):3319-29. PMID: 15132537.
Lee S-H, Matsushita H, Clapham B, Janda KD. The direct conversion of carbamates to ureas using aluminum amides. Tetrahedron. 2004;60(15):3439-43.
Lee SH, Yoshida K, Matsushita H, Clapham B, Koch G, Zimmermann J, Janda KD. N-H insertion reactions of primary ureas: The synthesis of highly substituted imidazolones and imidazoles from diazocarbonyls. J Org Chem. 2004;69(25):8829-35. PMID: 15575764.
Matsushita H, Lee SH, Yoshida K, Clapham B, Koch G, Zimmermann J, Janda KD. N-H insertion reactions of Boc-amino acid amides: Solution- and solid-phase synthesis of pyrazinones and pyrazines. Org Lett. 2004;6(24):4627-9. PMID: 15548092.
Matsushita H, Lee S-H, Joung M, Clapham B, Janda KD. Smart cleavage reactions: The synthesis of benzimidazoles and benzothiazoles from polymer-bound esters. Tetrahedron Lett. 2004;45(2):313-6.
Meijler MM, Hom LG, Kaufmann GF, McKenzie KM, Sun C, Moss JA, Matsushita M, Janda KD. Synthesis and biological validation of a ubiquitous quorum-sensing molecule. Angew Chem Int Ed Engl. 2004;43(16):2106-8. PMID: 15083457.
Qi L, Meijler MM, Lee SH, Sun C, Janda KD. Solid-phase synthesis of anandamide analogues. Org Lett. 2004;6(10):1673-5. PMID: 15128264.
Chen Y, Gambs C, Abe Y, Wentworth P, Jr., Janda KD. Total synthesis of the depsipeptide FR-901375. J Org Chem. 2003;68(23):8902-5. PMID: 14604360.
Dickerson TJ, Reed NN, Janda KD. Soluble polymers as catalyst and reagent platforms: Liquid-phase methodologies. In: Buchmeiser MR, editor. Polymeric Materials in Organic Synthesis and Catalysis. Weinheim, Germany: Wiley-VCH Verlag Gmbh; 2003. p. 241-76.
Lee SH, Clapham B, Koch G, Zimmermann J, Janda KD. Rhodium carbenoid N-H insertion reactions of primary ureas: Solution and solid-phase synthesis of imidazolones. Org Lett. 2003;5(4):511-4. PMID: 12583756.
Ahn JM, Boyle NA, MacDonald MT, Janda KD. Peptidomimetics and peptide backbone modifications. Mini Rev Med Chem. 2002;2(5):463-73. PMID: 12370047.
Boyle NA, Janda KD. Formats for combinatorial synthesis: Solid-phase, liquid-phase and surface. Curr Opin Chem Biol. 2002;6(3):339-46. PMID: 12023115.
Clapham B, Lee S-H, Koch G, Zimmermann J, Janda KD. The preparation of polymer bound β-ketoesters and their conversion into an array of oxazoles. Tetrahedron Lett. 2002;43(31):5407-10.
Delgado M, Janda KD. Polymeric supports for solid phase organic synthesis. Curr Org Chem. 2002;6(12):1031-43.
Delgado M, Spanka C, Kerwin LD, Wentworth P, Jr., Janda KD. A tunable hydrogel for encapsulation and controlled release of bioactive proteins. Biomacromolecules. 2002;3(2):262-71. PMID: 11888310.
Dickerson TJ, Janda KD. Aqueous aldol catalysis by a nicotine metabolite. J Am Chem Soc. 2002;124(13):3220-1. PMID: 11916401.
Dickerson TJ, Reed NN, Janda KD. Soluble polymers as scaffolds for recoverable catalysts and reagents. Chem Rev. 2002;102(10):3325-44. PMID: 12371887.
Isomura S, Ashley JA, Wirsching P, Janda KD. Antibody-catalyzed cleavage of the D-Ala-D-Lac depsipeptide: An immunological approach to the problem of vancomycin resistance. Bioorg Med Chem Lett. 2002;12(6):861-4. PMID: 11958980.
Isomura S, Hoffman TZ, Wirsching P, Janda KD. Synthesis, properties, and reactivity of cocaine benzoylthio ester possessing the cocaine absolute configuration. J Am Chem Soc. 2002;124(14):3661-8. PMID: 11929256.
Janda K. Polymer supported catalysts and reagents in synthetic organic chemistry. Bioorg Med Chem Lett. 2002;12(14):viii.
Kim GT, Wenz M, Park JI, Hasserodt J, Janda KD. Polyene substrates with unusual methylation patterns to probe the active sites of three catalytic antibodies. Bioorg Med Chem. 2002;10(5):1249-62. PMID: 11886788.
Matsushita M, Janda KD. Histidine kinases as targets for new antimicrobial agents. Bioorg Med Chem. 2002;10(4):855-67. PMID: 11836091.
Moss JA, Dickerson TJ, Janda KD. Solid phase peptide synthesis on JandaJelTM resin. Tetrahedron Lett. 2002;43(1):37-40.
Nicholas KM, Wentworth P, Jr., Harwig CW, Wentworth AD, Shafton A, Janda KD. A cofactor approach to copper-dependent catalytic antibodies. Proc Natl Acad Sci U S A. 2002;99(5):2648-53. PMID: 11880619.
Reger TS, Janda KD. Parallel suspension polymerization for high-throughput resin synthesis. Bioorg Med Chem Lett. 2002;12(6):837-40. PMID: 11958974.
Spanka C, Clapham B, Janda KD. Preparation of new microgel polymers and their application as supports in organic synthesis. J Org Chem. 2002;67(9):3045-50. PMID: 11975565.
Sun C, Wirsching P, Janda KD. Syntheses of dendritic linkers containing chlorambucil residues for the preparation of antibody-multidrug immunoconjugates. Bioorg Med Chem Lett. 2002;12(16):2213-5. PMID: 12127540.
Brümmer O, Clapham B, Janda KD. Solid-phase synthesis of oligoesters using a JandaJel™ resin. Tetrahedron Lett. 2001;42(12):2257-9.
Clapham B, Cho CW, Janda KD. A polymer-supported proline-based diamine catalyst for the kinetic resolution of racemic secondary alcohols. J Org Chem. 2001;66(3):868-73. PMID: 11430106.
Clapham B, Reger TS, Janda KD. Polymer-supported catalysis in synthetic organic chemistry. Tetrahedron. 2001;57(22):4637-62.
Córdova A, Janda KD. A highly chemo- and stereoselective synthesis of of β-keto esters via a polymer-supported lipase catalyzed transesterfication. J Org Chem. 2001;66(5):1906-9. PMID: 11262145.
Córdova A, Tremblay MR, Clapham B, Janda KD. A sequential application of kinetic resolution and polymer-supported scavenging for the isolation of chiral secondary alcohols. J Org Chem. 2001;66(16):5645-8. PMID: 11485501.
Lee KJ, Janda KD. Traceless solid-phase synthesis of 5-benzoylbenzimidazoles. Can J Chem. 2001;79(11):1556-61.
Wen K, Han H, Hoffman TZ, Janda KD, Orgel LE. The synthesis of β-peptides containing guanidino groups. Bioorg Med Chem Lett. 2001;11(5):689-91. PMID: 11266170.
Brümmer O, Clapham B, Janda KD. Recent developments and applications of polymer-supported reagents in synthetic organic chemistry. Curr Opin Drug Discov Devel. 2000;3(4):462-73. PMID: 19649877.
Harwig CW, Hoffman TZ, Wentworth AD, Janda KD. A one-pot multistep approach to alpha-azido-phosphonate and phosphonothioate diesters: Key intermediates in the synthesis of haptens for the generation of antibody ligases. Bioorg Med Chem Lett. 2000;10(9):915-8. PMID: 10853659.
Hasserodt J, Janda KD, Lerner RA. Antibodies mimic natural oxidosqualene−cyclase action in steroid ring a formation. J Am Chem Soc. 2000;122(1):40-5.
Lopez-Pelegrin JA, Janda KD. Solution- and soluble-polymer supported asymmetric syntheses of six-membered ring prostanoids. Chem Eur J. 2000;6(11):1917-22. PMID: 10894390.
Manzotti R, Reger TS, Janda KD. Improved synthesis of (4-ethenylphenyl)diphenyl methanol and its application in the preparation of trityl functionalized polystyrene resin containing tetrahydrofuran derived cross-linker. Tetrahedron Lett. 2000;41(44):8417-20.
Manzotti R, Tang S-Y, Janda KD. Improved synthesis of prostanoids on a non-cross-linked polystyrene soluble support. Tetrahedron. 2000;56(40):7885-92.
Reed NN, Janda KD. A one-step synthesis of monoprotected polyethylene glycol ethers. J Org Chem. 2000;65(18):5843-5. PMID: 10970334.
Reger TS, Janda KD. Polymer-supported (salen)Mn catalysts for asymmetric epoxidation: A comparison between soluble and insoluble matrices. J Am Chem Soc. 2000;122(29):6929-34.
Sieber F, Wentworth P, Janda KD. Exploiting poly(ethylene glycol) as a matrix for liquid-phase organic synthesis. Molecules. 2000;5(8):1018-32.
Toy PH, Janda KD. Soluble polymer-supported organic synthesis. Acc Chem Res. 2000;33(8):546-54. PMID: 10955985.
Toy PH, Reger TS, Janda KD. Soluble polymer bound cleavage reagents: A multipolymer strategy for the cleavage of tertiary amines from REM resin. Org Lett. 2000;2(15):2205-7. PMID: 10930244.
Tremblay MR, Wentworth P, Jr., Lee GE, Jr., Janda KD. Parallel solid-phase synthesis and structural characterization of a library of highly substituted chiral 1,3-oxazolidines. J Comb Chem. 2000;2(6):698-709. PMID: 11126298.
Vaino AR, Janda KD. Solid-phase organic synthesis: A critical understanding of the resin. J Comb Chem. 2000;2(6):579-96. PMID: 11126287.
Wentworth AD, Wentworth P, Jr., Mansoor UF, Janda KD. A soluble polymer-supported triflating reagent: A high-throughput synthetic approach to aryl and enol triflates. Org Lett. 2000;2(4):477-80. PMID: 10814355.
Berg T, Simeonov A, Janda KD. A combined parallel synthesis and screening of macrocyclic lanthanide complexes for the cleavage of phospho di- and triesters and double-stranded DNA. J Comb Chem. 1999;1(1):96-100. PMID: 10746017.
Brümmer O, Wentworth P, Weiner DP, Janda KD. Phosphorodithioates: Synthesis and evaluation of new haptens for the generation of antibody acyl transferases. Tetrahedron Lett. 1999;40(41):7307-10.
Córdova A, Reed NN, Ashley JA, Janda KD. Convenient synthesis of L-proline benzyl ester. Bioorg Med Chem Lett. 1999;9(21):3119-22. PMID: 10560736.
Han H, Cho C-W, Janda KD. A substrate‐based methodology that allows the regioselective control of the catalytic aminohydroxylation reaction. Chemistry: A European Journal. 1999;5:1565-9.
Lee KJ, Angulo A, Ghazal P, Janda KD. Soluble-polymer supported synthesis of a prostanoid library: Identification of antiviral activity. Org Lett. 1999;1(11):1859-62. PMID: 10836045.
Wentworth Jr P, D. Janda K. Liquid-phase chemistry: Recent advances in soluble polymer-supported catalysts, reagents and synthesis. Chem Commun. 1999;10.1039/A901955C(19):1917-24.
Chen S, Janda KD. Total synthesis of naturally occurring prostaglandin F2α on a non-cross-linked polystyrene support. Tetrahedron Lett. 1998;39(23):3943-6.
Gravert DJ, Janda KD. Bifunctional initiators for free radical polymerization of non-crosslinked block copolymers. Tetrahedron Lett. 1998;39(12):1513-6.
Han H, Yoon J, Janda KD. An efficient asymmetric route to 2,3-ciaminobutanoic acids. J Org Chem. 1998;63(6):2045-8.
Hori M, Janda KD. A soluble polymer approach to the “fishing out" principle: Synthesis and purification of -amino alcohols. J Org Chem. 1998;63(3):889-94. PMID: 11672090.
Yli-Kauhaluoma JT, Harwig CW, Wentworth P, Janda KD. Unexpected 1,3-oxazolidine formation in the attempted oxidation of N-aryl-N-methyl substituted β-amino alcohols using pyridinium dichromate. Tetrahedron Lett. 1998;39(16):2269-72.
Yoon J, Cho C-W, Han H, D. Janda K. Solution and soluble polymer syntheses of 3-aminoimidazoline-2,4-diones. Chem Commun. 1998;10.1039/A807067I(24):2703-4.
Chen S, Janda KD. Synthesis of prostaglandin E2 methyl ester on a soluble-polymer support for the construction of prostanoid libraries. J Am Chem Soc. 1997;119(37):8724-5.
Gravert DJ, Janda KD. Synthesis on soluble polymers: New reactions and the construction of small molecules. Curr Opin Chem Biol. 1997;1(1):107-13. PMID: 9667833.
Han H, Janda KD. A soluble polymer-bound approach to the Sharpless catalytic asymmetric dihydroxylation (AD) reaction: Preparation and application of a [(DHQD)2PHAL-PEG-OMe] ligand. Tetrahedron Lett. 1997;38(9):1527-30.
Han H, Janda KD. Multipolymer-supported substrate and ligand approach to the Sharpless asymmetric dihydroxylation. Angew Chem Int Ed Engl. 1997;36(16):1731-3.
Hasserodt J, Janda KD. Syntheses of octahydroquinoline-N-oxides: Haptens designed to elicit catalytic antibodies that control a terpenoid-like cascade cyclisation. Tetrahedron. 1997;53(33):11237-56.
Wentworth Jr P, Janda KD. Synthesis of oxorhenium (V) and oxotechnetium (V) complexes as inhibitors of ribonucleases and for the generation of catalytic antibodies. Synlett. 1997;1997(05):537-43.
Han H, Janda KD. Soluble polymer-bound ligand-accelerated catalysis: Asymmetric dihydroxylation. J Am Chem Soc. 1996;118(32):7632-3.
Han H, Janda KD. Azatides: Solution and liquid phase syntheses of a new peptidomimetic. J Am Chem Soc. 1996;118(11):2539-44.
Jung KW, Janda KD, Sanfilippo PJ, Wachter M. Syntheses and biological evaluation of two new naproxen analogs. Bioorg Med Chem Lett. 1996;6(19):2281-2.
Sakurai M, Wirsching P, Janda KD. Design and synthesis of a cocaine-diamide hapten for vaccine development. Tetrahedron Lett. 1996;37(31):5479-82.
Sakurai M, Wirsching P, Janda KD. Synthesis of a nucleoside hapten with a [P(O)-O-N] linkage to elicit catalytic antibodies with phosphodiesterase activity. Bioorg Med Chem Lett. 1996;6(9):1055-60.
Wentworth P, Janda KD. A facile and efficient route to 3′,5′-diamino-3′,5′-dideoxynucleosides. Chem Commun. 1996;10.1039/CC9960002097(17):2097-8.
Wentworth P, Wiemann T, Janda KD. A new class of pentacoordinate ribonuclease inhibitors: Synthesis, characterization, and inhibition studies of ribonucleoside and anhydropentofuranose oxorhenium(V) complexes. J Am Chem Soc. 1996;118(50):12521-7.
Lavey BJ, Janda KD. Applying antibody catalysis to organic synthesis. In: Wang HY, Imanaka T, editors. Antibody Expression and Engineering (ACS Symposium Series, No 604). 1st ed: American Chemical Society; 1995. p. 123.
Shevlin CG, Hilton S, Janda KD. Automation of antibody catalysis: A practical methodology for the use of catalytic antibodies in organic synthesis. Bioorg Med Chem Lett. 1994;4(2):297-302.
Yli-Kauhaluoma J, Janda KD. Twisted α-keto amides as transition-state analogues for acyl-transfer reactions: Synthesis of the immunoconjugates. Bioorg Med Chem. 1994;2(6):521-8. PMID: 7528089.
Yli-Kauhaluoma JT, Janda KD. An expedient synthesis of isopropyl anisoles and veratroles. Tetrahedron Lett. 1994;35(26):4509-10.
Janda KD. Book review on “Studies in organic chemistry. 46. Biocatalysts in organic synthesis” by J. Halgas. J Am Chem Soc. 1993;115(19):8888-9.
Weinhouse MI, Janda KD. A new methodology for the preparation of vinyl esters. Synthesis. 1993;1993(1):81-3.
Chen YCJ, Janda KD. A new approach toward the inhibition of ribonucleases: A water-stable ribonucleoside-technetium chelate. J Am Chem Soc. 1992;114(4):1488-9.
Ikeda S, Ashley JA, Wirsching P, Janda KD. ψ[PO2-CH2N+], a new amide bond replacement: Potent, slow-binding inhibition of the HIV protease. J Am Chem Soc. 1992;114(19):7604-6.
Chen YCJ, Hansske F, Janda KD, Robins MJ. Nucleic acid related compounds. 64. Synthesis of 2',3'-diazido-2',3'-dideoxyadenosine and 2',3'-diamino-2',3'-dideoxyadenosine from 9-(β-D-arabinofuranosyl)adenine. J Org Chem. 1991;56(10):3410-3.
Janda KD. Opportunities in organic synthesis for catalytic antibodies. Proceedings of 15th ABC Symposium, Kyoto, Japan. 1991;3:63.
McLeod DA, Brinkworth RI, Ashley JA, Janda KD, Wirsching P. Phosphonamidates and phosphonamidate esters as HIV-1 protease inhibitors. Bioorg Med Chem Lett. 1991;1(11):653-8.
Janda KD, Ashley JA. Syntheses of the saturated analogues of 4-nitrophenol and 4-nitroaniline. Synth Commun. 1990;20(7):1073-82.
Bates RB, Janda KD, Wright ME. N-Isobutyrylbenzamide, C11H13NO2. Acta Crystallogr C: Struct Chem. 1985;C41(2):263-4.
Bates RB, Fletcher FA, Janda KD, Miller WA. A convenient synthesis of unsymmetrical acyclic imides. J Org Chem. 1984;49(16):3038.
Bates RB, Gin SL, Hassen MA, Hruby VJ, Janda KD, Kriek GR, Michaud J-P, Vine DB. Synthesis of cyclo-N-methyl-L-tyr-N-methyl-L-tyr-D-ala-L-ala-O,N-dimethyl-L-tyr-L-ala, a cyclic hexapeptide related to the antitumor agent Deoxybouvardin. Heterocycles. 1984;22(4):785 - 90.
Bates RB, Janda KD. A convenient synthesis of α-acylamino alcohols from azlactones. Synthesis. 1984;1984(04):310-1.
Janda KD, McConnell WW, Nelson GO, Wright ME. Preparation and reactivity of the new cyclopentadienyl-bridged complex (Me2SiCH2CH2SiMe2)(C5H4Fe(CO)2)2. J Organomet Chem. 1983;259(2):139-43.
Bates RB, Janda KD. High-yield benzyne synthesis of diaryl ethers. J Org Chem. 1982;47(22):4374-6.
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